Fragment-based discovery of potent and selective DDR1/2 inhibitors

Fragment-based discovery of potent and selective DDR1/2 inhibitors Descriptor: Epithelial discoidin domain-containing receptor 1, IODIDE ION, N-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide Authors: Murray, C, Berdini, V, Buck, I, Carr, M, Cleasby, A, Coyle, J, Curry, J, Day, J, Hearn, K, Iqbal, A, Lee, L, Martins, V, Mortenson, P, Munck, J, Page, L, Patel, S, Roomans, S, Kirsten, T, Saxty, G. Deposit date: 2015-06-05 Release date: 2015-08-12 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.21 Å) Cite: Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors. Acs Med.Chem.Lett., 6, 2015