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Crystal structure of human DYRK1A in complex with ARN25068

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Protein Data Bank Japan2024-10-23 更新2026-03-28 收录
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Crystal structure of human DYRK1A in complex with ARN25068 Descriptor: Dual specificity tyrosine-phosphorylation-regulated kinase 1A, ~{N}4-(3-cyclopropyl-1~{H}-pyrazol-5-yl)-~{N}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamine Authors: Tripathi, S.K, Balboni, B, Demuro, S, DiMartino, R, Ortega, J, Girotto, S, Cavalli, A. Deposit date: 2021-06-23 Release date: 2022-03-02 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.38 Å) Cite: ARN25068, a versatile starting point towards triple GSK-3 beta /FYN/DYRK1A inhibitors to tackle tau-related neurological disorders. Eur.J.Med.Chem., 229, 2022
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2021-06-23
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