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BAZ2A bromodomain in complex with isoquinoline derivative fragment 9

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Protein Data Bank Japan2024-01-31 更新2026-04-19 收录
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资源简介:
BAZ2A bromodomain in complex with isoquinoline derivative fragment 9 Descriptor: Bromodomain adjacent to zinc finger domain protein 2A, ~{N}-[(3~{S})-pyrrolidin-3-yl]isoquinoline-5-sulfonamide Authors: Dalle Vedove, A, Cazzanelli, G, Caflisch, A, Lolli, G. Deposit date: 2022-01-31 Release date: 2022-09-28 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.183 Å) Cite: Identification of a BAZ2A-Bromodomain Hit Compound by Fragment Growing. Acs Med.Chem.Lett., 13, 2022
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2022-01-31
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