Ligand complex of RORg LBD
收藏Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Ligand complex of RORg LBD Descriptor: 2-CHLORO-6-FLUORO-N-[4-[3-(TRIFLUOROMETHYL)PHENYL]SULFONYL-3,5-DIHYDRO-2H-1,4-BENZOXAZEPIN-7-YL]BENZAMIDE, NUCLEAR RECEPTOR COACTIVATOR 2, NUCLEAR RECEPTOR ROR-GAMMA, ... Authors: Xue, Y, Aagaard, A, Narjes, F. Deposit date: 2015-09-16 Release date: 2015-11-25 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.08 Å) Cite: Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper 17 (TH 17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor ROR gamma. ChemMedChem, 11, 2016
创建时间:
2015-09-16



