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The Structure of CK2alpha with CCh507 bound

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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The Structure of CK2alpha with CCh507 bound Descriptor: ADENOSINE-5'-TRIPHOSPHATE, Casein kinase II subunit alpha, [1-[2-(phenylsulfonylamino)ethyl]piperidin-4-yl]methyl 1~{H}-indole-3-carboxylate Authors: Brear, P, Prudent, R, Laudet, B, Filhol, O, Cochet, C, Sautel, C, Moucadel, V, Bestgen, B, Engel, M, Ettaoussi, M, Lomberget, T, Le Borgne, M, Kufareva, I, Abagyan, R, Hyvonen, M. Deposit date: 2018-03-02 Release date: 2019-06-19 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.6 Å) Cite: Discovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitors. Sci Rep, 9, 2019
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2018-03-02
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