Crystal structure of E. coli HPPK in complex with bisubstrate analogue inhibitor J1A
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Crystal structure of E. coli HPPK in complex with bisubstrate analogue inhibitor J1A Descriptor: 1,2-ETHANEDIOL, 2-amino-4-hydroxy-6-hydroxymethyldihydropteridine pyrophosphokinase, 5'-S-[1-(2-{[(2-amino-4-oxo-3,4-dihydropteridin-6-yl)methyl]amino}ethyl)piperidin-4-yl]-5'-thioadenosine Authors: Shaw, G, Shi, G, Ji, X. Deposit date: 2011-10-27 Release date: 2012-01-04 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (2 Å) Cite: Bisubstrate analogue inhibitors of 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase: New design with improved properties. Bioorg.Med.Chem., 20, 2012
创建时间:
2011-10-27



