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Bromodomain-containing protein 4 (BRD4) bromodomain 2 (BD2) complexed with YF3-126

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Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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https://pdbj.org/mine/summary/7jkz
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资源简介:
Bromodomain-containing protein 4 (BRD4) bromodomain 2 (BD2) complexed with YF3-126 Descriptor: 1,2-ETHANEDIOL, Bromodomain-containing protein 4, GLYCEROL, ... Authors: Ratia, K.M, Xiong, R, Li, Y, Shen, Z, Zhao, J, Huang, F, Dubrovyskyii, O, Thatcher, G.R. Deposit date: 2020-07-29 Release date: 2021-08-25 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.49 Å) Cite: Novel Pyrrolopyridone Bromodomain and Extra-Terminal Motif (BET) Inhibitors Effective in Endocrine-Resistant ER+ Breast Cancer with Acquired Resistance to Fulvestrant and Palbociclib. J.Med.Chem., 63, 2020
创建时间:
2020-07-29
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