[1,2,4]Triazolo[1,5-a]pyrimidine Phosphodiesterase 2 Inhibitors
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[1,2,4]Triazolo[1,5-a]pyrimidine Phosphodiesterase 2 Inhibitors Descriptor: MAGNESIUM ION, ZINC ION, [(3~{S})-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]-(3,4,5-trimethoxyphenyl)methanone, ... Authors: Tresadern, G, Leonard, P.M. Deposit date: 2020-07-06 Release date: 2020-07-22 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.35 Å) Cite: [1,2,4]Triazolo[1,5- a ]pyrimidine Phosphodiesterase 2A Inhibitors: Structure and Free-Energy Perturbation-Guided Exploration. J.Med.Chem., 63, 2020
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2020-07-06



