IRAK4 in complex with a type II inhibitor
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IRAK4 in complex with a type II inhibitor Descriptor: 3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}-N-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide, COBALT (II) ION, Interleukin-1 receptor-associated kinase 4, ... Authors: Wang, L, Wu, H. Deposit date: 2018-08-19 Release date: 2019-02-20 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.512 Å) Cite: Conformational flexibility and inhibitor binding to unphosphorylated interleukin-1 receptor-associated kinase 4 (IRAK4). J.Biol.Chem., 294, 2019
创建时间:
2018-08-19



