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BAZ2A bromodomain in complex with acetylpyrrole derivative compound 113

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Protein Data Bank Japan2024-01-31 更新2026-04-19 收录
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BAZ2A bromodomain in complex with acetylpyrrole derivative compound 113 Descriptor: (2~{R})-~{N}-(2,2-dimethylpropyl)-1-[4-(4-ethanoyl-3-ethyl-5-methyl-1~{H}-pyrrol-2-yl)-1,3-thiazol-2-yl]piperazine-2-carboxamide, 1,2-ETHANEDIOL, Bromodomain adjacent to zinc finger domain protein 2A, ... Authors: Dalle Vedove, A, Cazzanelli, G, Caflisch, A, Lolli, G. Deposit date: 2022-01-31 Release date: 2022-09-28 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.98 Å) Cite: Identification of a BAZ2A-Bromodomain Hit Compound by Fragment Growing. Acs Med.Chem.Lett., 13, 2022

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2022-01-31
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