p38alpha in complex with pyrazolobenzothiazine inhibitor COXP4M12
收藏Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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p38alpha in complex with pyrazolobenzothiazine inhibitor COXP4M12 Descriptor: 3-(4-fluorophenyl)-4-methyl-1~{H}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide, Mitogen-activated protein kinase 14, octyl beta-D-glucopyranoside Authors: Buehrmann, M, Rauh, D. Deposit date: 2017-07-31 Release date: 2019-03-13 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2 Å) Cite: Co-crystal structure determination and cellular evaluation of 1,4-dihydropyrazolo[4,3-c] [1,2] benzothiazine 5,5-dioxide p38 alpha MAPK inhibitors. Biochem.Biophys.Res.Commun., 511, 2019
创建时间:
2017-07-31



