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tRNA-guanine Transglycosylase (TGT) in complex with 6-Amino-4-[2-(4-methylphenyl)ethyl]-1,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one

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Protein Data Bank Japan2023-10-25 更新2026-03-21 收录
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https://pdbj.org/mine/summary/1y5w
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资源简介:
tRNA-guanine Transglycosylase (TGT) in complex with 6-Amino-4-[2-(4-methylphenyl)ethyl]-1,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one Descriptor: 6-AMINO-4-[2-(4-METHYLPHENYL)ETHYL]-1,7-DIHYDRO-8H-IMIDAZO[4,5-G]QUINAZOLIN-8-ONE, GLYCEROL, Queuine tRNA-ribosyltransferase, ... Authors: Stengl, B, Meyer, E.A, Heine, A, Brenk, R, Diederich, F, Klebe, G. Deposit date: 2004-12-03 Release date: 2005-12-13 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.58 Å) Cite: Crystal structures of tRNA-guanine transglycosylase (TGT) in complex with novel and potent inhibitors unravel pronounced induced-fit adaptations and suggest dimer formation upon substrate binding J.Mol.Biol., 370, 2007
创建时间:
2004-12-03
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