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CDK1/Cks2 in complex with Dinaciclib

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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CDK1/Cks2 in complex with Dinaciclib Descriptor: 3-[({3-ethyl-5-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium, Cyclin-dependent kinase 1, Cyclin-dependent kinases regulatory subunit 2 Authors: Wood, D.J, Korolchuk, S, Tatum, N.J, Wang, L.Z, Endicott, J.A, Noble, M.E.M, Martin, M.P. Deposit date: 2018-06-19 Release date: 2018-12-05 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (2.33 Å) Cite: Differences in the Conformational Energy Landscape of CDK1 and CDK2 Suggest a Mechanism for Achieving Selective CDK Inhibition. Cell Chem Biol, 26, 2019
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2018-06-19
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