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Hsp90 Alpha N-terminal Domain in Complex with an Inhibitor 3-(4-Hydroxy-phenyl)-1H-indazol-6-ol

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Protein Data Bank Japan2024-03-20 更新2026-03-21 收录
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Hsp90 Alpha N-terminal Domain in Complex with an Inhibitor 3-(4-Hydroxy-phenyl)-1H-indazol-6-ol Descriptor: 3-(4-hydroxyphenyl)-1H-indazol-6-ol, Heat shock protein HSP 90-alpha, SULFATE ION Authors: Musil, D, Lehmann, M, Graedler, U, Buchstaller, H.-P. Deposit date: 2012-03-28 Release date: 2012-06-27 Last modified: 2024-03-20 Method: X-RAY DIFFRACTION (1.6 Å) Cite: Fragment-based discovery of hydroxy-indazole-carboxamides as novel small molecule inhibitors of Hsp90 Bioorg.Med.Chem.Lett., 22, 2012

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2012-03-28
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