five

Murine PI3K delta kinsae domain - cpd 1

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6mul
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资源简介:
Murine PI3K delta kinsae domain - cpd 1 Descriptor: 1-{1-[8-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-9-methyl-9H-purin-6-yl]piperidin-4-yl}-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform Authors: Fischmann, T.O. Deposit date: 2018-10-23 Release date: 2019-05-01 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (3.09 Å) Cite: Structure Overhaul Affords a Potent Purine PI3K delta Inhibitor with Improved Tolerability. J.Med.Chem., 62, 2019
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2018-10-23
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