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Tubulin Polymerization Inhibitors

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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Tubulin Polymerization Inhibitors Descriptor: 2-(4-methylphenyl)-7-(3,4,5-trimethoxyphenyl)pyrazolo[1,5-a]pyrimidine, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ... Authors: Gang, L, Wang, Y.X, Chen, J.J. Deposit date: 2020-01-17 Release date: 2021-01-20 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.751 Å) Cite: Design, Synthesis, and Bioevaluation of Pyrazolo[1,5-a]Pyrimidine Derivatives as Tubulin Polymerization Inhibitors Targeting the Colchicine Binding Site with Potent Anticancer Activities To Be Published

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2020-01-17
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