Structure of protein kinase ck2 catalytic subunit (csnk2a2 gene product) in complex with the bivalent inhibitor KN2
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Structure of protein kinase ck2 catalytic subunit (csnk2a2 gene product) in complex with the bivalent inhibitor KN2 Descriptor: 1,2-ETHANEDIOL, CHLORIDE ION, Casein kinase II subunit alpha', ... Authors: Lindenblatt, D, Applegate, V, Nickelsen, A, Klussmann, M, Neundorf, I, Goetz, C, Jose, J, Niefind, K. Deposit date: 2020-10-31 Release date: 2021-08-04 Last modified: 2024-06-19 Method: X-RAY DIFFRACTION (0.98 Å) Cite: Molecular Plasticity of Crystalline CK2 alpha ' Leads to KN2, a Bivalent Inhibitor of Protein Kinase CK2 with Extraordinary Selectivity. J.Med.Chem., 65, 2022
创建时间:
2020-10-31



