遇见数据集

First bromodomain of BRD4 liganded with CCS-1477

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Protein Data Bank Japan2024-06-05 更新2026-04-19 收录
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First bromodomain of BRD4 liganded with CCS-1477 Descriptor: (6S)-1-[3,4-bis(fluoranyl)phenyl]-6-[5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-(4-methoxycyclohexyl)benzimidazol-2-yl]piperidin-2-one, 1,2-ETHANEDIOL, Bromodomain-containing protein 4 Authors: Schonbrunn, E, Bikowitz, M. Deposit date: 2023-01-19 Release date: 2024-02-07 Last modified: 2024-06-05 Method: X-RAY DIFFRACTION (1.53 Å) Cite: Group 3 medulloblastoma transcriptional networks collapse under domain specific EP300/CBP inhibition. Nat Commun, 15, 2024

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2023-01-19
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