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Human MALT1(329-729) in complex with a chromane urea containing inhibitor

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Protein Data Bank Japan2024-01-31 更新2026-03-21 收录
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Human MALT1(329-729) in complex with a chromane urea containing inhibitor Descriptor: 1-[4-[4-(aminomethyl)pyrazol-1-yl]-3-chloranyl-phenyl]-3-[(3~{R})-6-bromanyl-3,4-dihydro-2~{H}-chromen-3-yl]urea, Mucosa-associated lymphoid tissue lymphoma translocation protein 1 Authors: Renatus, M. Deposit date: 2020-09-29 Release date: 2020-12-09 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.316 Å) Cite: Discovery of Potent, Highly Selective, and In Vivo Efficacious, Allosteric MALT1 Inhibitors by Iterative Scaffold Morphing. J.Med.Chem., 63, 2020
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2020-09-29
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