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Structure of liver pyruvate kinase in complex with Liver pyruvate kinase in complex with fluorescent probe I

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Protein Data Bank Japan2026-04-15 更新2026-08-24 收录
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Structure of liver pyruvate kinase in complex with Liver pyruvate kinase in complex with fluorescent probe I Descriptor: 1,6-di-O-phosphono-beta-D-fructofuranose, 2-(phenylmethyl)-6-(phenylsulfonyl)phthalazin-1-one, Isoform L-type of Pyruvate kinase PKLR, ... Authors: Bogucka, A, Koteles, I, Grotli, M, Hyvonen, M. Deposit date: 2025-06-04 Release date: 2026-04-08 Last modified: 2026-04-15 Method: X-RAY DIFFRACTION (2.385 Å) Cite: Potent Fluorescent Probe for Target-Engagement Studies of Allosteric Pyruvate Kinase Modulators. Angew.Chem.Int.Ed.Engl., 64, 2025

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2025-06-04
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