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C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 2-benzyl-N-cyclopropyl-6-(1-methyl-1H-1,2,3-triazol-4-yl)isonicotinamide

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Protein Data Bank Japan2024-06-19 更新2026-03-21 收录
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https://pdbj.org/mine/summary/7nqi
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C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 2-benzyl-N-cyclopropyl-6-(1-methyl-1H-1,2,3-triazol-4-yl)isonicotinamide Descriptor: 1,2-ETHANEDIOL, 2-benzyl-N-cyclopropyl-6-(1-methyl-1H-1,2,3-triazol-4-yl)isonicotinamide, Bromodomain-containing protein 2 Authors: Chung, C.W. Deposit date: 2021-03-01 Release date: 2021-03-24 Last modified: 2024-06-19 Method: X-RAY DIFFRACTION (1.603 Å) Cite: Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors. J.Med.Chem., 64, 2021
创建时间:
2021-03-01
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