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Crystal structure of PI3K-gamma in complex with quinoline-indoline inhibitor 24f

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Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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Crystal structure of PI3K-gamma in complex with quinoline-indoline inhibitor 24f Descriptor: 4-[3,3-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1H-indol-1-yl]-7-fluoro-3-methyl-2-(pyridin-3-yl)quinoline, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION Authors: Whittington, D.A, Tang, J, Yakowec, P. Deposit date: 2012-06-12 Release date: 2012-10-24 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (2.9 Å) Cite: Discovery and in Vivo Evaluation of Dual PI3K-beta/delta inhibitors J.Med.Chem., 55, 2012
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2012-06-12
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