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Crystal structure of the Mycobacterium tuberculosis PknB mutant kinase domain in complex with KT5720

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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https://pdbj.org/mine/summary/3f69
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Crystal structure of the Mycobacterium tuberculosis PknB mutant kinase domain in complex with KT5720 Descriptor: SULFATE ION, Serine/threonine-protein kinase pknB, hexyl (5S,6R,8R)-6-hydroxy-5-methyl-13-oxo-5,6,7,8-tetrahydro-13H-5,8-epoxy-4b,8a,14-triazadibenzo[b,h]cycloocta[1,2,3,4-jkl]c yclopenta[e]-as-indacene-6-carboxylate Authors: Alber, T, Mieczkowski, C.A, TB Structural Genomics Consortium (TBSGC) Deposit date: 2008-11-05 Release date: 2008-12-02 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.8 Å) Cite: Auto-activation mechanism of the Mycobacterium tuberculosis PknB receptor Ser/Thr kinase. Embo J., 27, 2008
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2008-11-05
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