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IRE1 kinase/RNase in complex with imidazo[1,2-b]pyridazin-8-amine compound 33

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6hv0
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资源简介:
IRE1 kinase/RNase in complex with imidazo[1,2-b]pyridazin-8-amine compound 33 Descriptor: 6-chloranyl-3-(2~{H}-indazol-5-yl)-~{N}-propan-2-yl-imidazo[1,2-b]pyridazin-8-amine, Serine/threonine-protein kinase/endoribonuclease IRE1 Authors: Bayliss, R, Bhatia, C, Collins, I. Deposit date: 2018-10-09 Release date: 2019-02-27 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.73 Å) Cite: Binding to an Unusual Inactive Kinase Conformation by Highly Selective Inhibitors of Inositol-Requiring Enzyme 1 alpha Kinase-Endoribonuclease. J.Med.Chem., 62, 2019
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2018-10-09
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