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Human MALT1(329-729) in complex with a chromane urea containing inhibitor

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Protein Data Bank Japan2024-01-31 更新2026-03-21 收录
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https://pdbj.org/mine/summary/7ak1
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Human MALT1(329-729) in complex with a chromane urea containing inhibitor Descriptor: 1-(3-chloranyl-4-methoxy-phenyl)-3-[7-[(3~{S})-3-(methoxymethyl)morpholin-4-yl]-2-methyl-pyrazolo[1,5-a]pyrimidin-6-yl]urea, MAGNESIUM ION, Mucosa-associated lymphoid tissue lymphoma translocation protein 1 Authors: Renatus, M. Deposit date: 2020-09-29 Release date: 2020-12-09 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.507 Å) Cite: Discovery of Potent, Highly Selective, and In Vivo Efficacious, Allosteric MALT1 Inhibitors by Iterative Scaffold Morphing. J.Med.Chem., 63, 2020
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2020-09-29
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