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TRPC4 in complex with inhibitor GFB-8749

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Protein Data Bank Japan2024-05-01 更新2026-03-21 收录
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TRPC4 in complex with inhibitor GFB-8749 Descriptor: (2R)-3-(phosphonooxy)propane-1,2-diyl dihexanoate, 4-[4-[[4,4-bis(fluoranyl)cyclohexyl]methyl]-3-oxidanylidene-piperazin-1-yl]-5-chloranyl-1~{H}-pyridazin-6-one, CALCIUM ION, ... Authors: Vinayagam, D, Quentin, D, Sistel, O, Merino, F, Stabrin, M, Hofnagel, O, Ledeboer, M.W, Malojcic, G, Raunser, S. Deposit date: 2020-11-18 Release date: 2020-12-09 Last modified: 2024-05-01 Method: ELECTRON MICROSCOPY (3.8 Å) Cite: Structural basis of TRPC4 regulation by calmodulin and pharmacological agents. Elife, 9, 2020

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2020-11-18
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