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Cryo-EM structure of the P395-bound GPBAR-Gs complex

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Protein Data Bank Japan2024-10-09 更新2026-03-21 收录
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Cryo-EM structure of the P395-bound GPBAR-Gs complex Descriptor: 2-(ethylamino)-6-[3-(4-propan-2-ylphenyl)propanoyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-4-carboxamide, CHOLESTEROL, G-protein coupled bile acid receptor 1, ... Authors: Yang, F, Mao, C, Guo, L, Lin, J, Ming, Q, Xiao, P, Wu, X, Shen, Q, Guo, S, Shen, D, Lu, R, Zhang, L, Huang, S, Ping, Y, Zhang, C, Ma, C, Zhang, K, Liang, X, Shen, Y, Nan, F, Yi, F, Luca, V, Zhou, J, Jiang, C, Sun, J, Xie, X, Yu, X, Zhang, Y. Deposit date: 2020-06-27 Release date: 2020-09-09 Last modified: 2024-10-09 Method: ELECTRON MICROSCOPY (3 Å) Cite: Structural basis of GPBAR activation and bile acid recognition. Nature, 587, 2020

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2020-06-27
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