MerTK kinase domain with type 1.5 inhibitor containing a tri-methyl pyrazole group
收藏Protein Data Bank Japan2024-01-31 更新2026-03-28 收录
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https://pdbj.org/mine/summary/7olx
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MerTK kinase domain with type 1.5 inhibitor containing a tri-methyl pyrazole group Descriptor: CHLORIDE ION, Tyrosine-protein kinase Mer, ~{N}-[[3-[4-[(dimethylamino)methyl]phenyl]imidazo[1,2-a]pyridin-6-yl]methyl]-~{N}-methyl-5-[3-methyl-5-(1,3,5-trimethylpyrazol-4-yl)pyridin-2-yl]-1,3,4-oxadiazol-2-amine Authors: Pflug, A, Schimpl, M, McCoull, W, Nissink, J.W.M, Winter-Holt, J. Deposit date: 2021-05-20 Release date: 2021-09-15 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.98 Å) Cite: Optimization of an Imidazo[1,2- a ]pyridine Series to Afford Highly Selective Type I1/2 Dual Mer/Axl Kinase Inhibitors with In Vivo Efficacy. J.Med.Chem., 64, 2021
创建时间：
2021-05-20
