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Structure of human PDK1 kinase domain in complex with LY333531

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Structure of human PDK1 kinase domain in complex with LY333531 Descriptor: (9R)-9-[(DIMETHYLAMINO)METHYL]-6,7,10,11-TETRAHYDRO-9H,18H-5,21:12,17-DIMETHENODIBENZO[E,K]PYRROLO[3,4-H][1,4,13]OXADIA ZACYCLOHEXADECINE-18,20-DIONE, 3-PHOSPHOINOSITIDE DEPENDENT PROTEIN KINASE-1, GLYCEROL, ... Authors: Komander, D, Kular, G.S, Schuttelkopf, A.W, Deak, M, Prakash, K.R, Bain, J, Elliot, M, Garrido-Franco, M, Kozikowski, A.P, Alessi, D.R, Van Aalten, D.M.F. Deposit date: 2003-12-15 Release date: 2004-03-04 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.7 Å) Cite: Interactions of Ly333531 and Other Bisindolyl Maleimide Inhibitors with Pdk1 Structure, 12, 2004

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2003-12-15
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