Mtb TMK in complex with compound 23
收藏Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4unr
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Mtb TMK in complex with compound 23 Descriptor: 4-[3-cyano-2-oxo-7-(1H-pyrazol-4-yl)-5,6-dihydro-1H-benzo[h]quinolin-4-yl]benzoic acid, MAGNESIUM ION, Thymidylate kinase Authors: Read, J.A, Hussein, S, Gingell, H, Tucker, J. Deposit date: 2014-05-30 Release date: 2015-06-17 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.98 Å) Cite: Structure Guided Lead Generation for M. Tuberculosis Thymidylate Kinase (Mtb Tmk): Discovery of 3-Cyanopyridone and 1,6-Naphthyridin-2-One as Potent Inhibitors. J.Med.Chem., 58, 2015
创建时间:
2014-05-30



