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Crystal structure of HIV-1 reverse transcriptase (RT) in complex with JANSSEN-R165481

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Protein Data Bank Japan2023-08-23 更新2026-03-21 收录
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Crystal structure of HIV-1 reverse transcriptase (RT) in complex with JANSSEN-R165481 Descriptor: (2E)-3-{3-[(5-ETHYL-3-IODO-6-METHYL-2-OXO-1,2-DIHYDROPYRIDIN-4-YL)OXY]PHENYL}ACRYLONITRILE, MANGANESE (II) ION, Reverse transcriptase P51 SUBUNIT, ... Authors: Himmel, D.H, Das, K, Clark Jr, A.D, Hughes, S.H, Benjahad, A, Oumouch, S, Guillemont, J, Coupa, S, Poncelet, A, Csoka, I, Meyer, C, Andries, K, Mguyen, C.H, Grierson, D.S, Arnold, E. Deposit date: 2005-09-28 Release date: 2005-12-06 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (2.9 Å) Cite: Crystal Structures for HIV-1 Reverse Transcriptase in Complexes with Three Pyridinone Derivatives: A New Class of Non-Nucleoside Inhibitors Effective against a Broad Range of Drug-Resistant Strains. J.Med.Chem., 48, 2005
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2005-09-28
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