five

BRD4 Bromodomain 1 in complex with multi-action inhibitor SF2523P

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Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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BRD4 Bromodomain 1 in complex with multi-action inhibitor SF2523P Descriptor: 3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(piperazin-1-yl)-7H-thieno[3,2-b]pyran-7-one, Bromodomain-containing protein 4 Authors: Vann, K.R, Kutateladze, T.G. Deposit date: 2020-05-29 Release date: 2020-08-05 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.5 Å) Cite: Design of thienopyranone-based BET inhibitors that bind multiple synthetic lethality targets. Sci Rep, 10, 2020
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2020-05-29
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