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Calpain 1 proteolytic core inactivated by WR18(S,S), an epoxysuccinyl-type inhibitor.

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2nqg
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资源简介:
Calpain 1 proteolytic core inactivated by WR18(S,S), an epoxysuccinyl-type inhibitor. Descriptor: 5-AZANYLIDYNE-N-[(2S)-4-ETHOXY-2-HYDROXY-4-OXOBUTANOYL]-L-NORVALYL-L-ARGINYL-L-TRYPTOPHANAMIDE, CALCIUM ION, Calpain-1 catalytic subunit Authors: Cuerrier, D, Davies, P.L, Campbell, R.L, Moldoveanu, T. Deposit date: 2006-10-31 Release date: 2007-01-09 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.04 Å) Cite: Development of Calpain-specific Inactivators by Screening of Positional Scanning Epoxide Libraries J.Biol.Chem., 282, 2007
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2006-10-31
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