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CRYSTAL STRUCTURE OF BACE-1 IN COMPLEX WITH CHEMICAL LIGAND

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF BACE-1 IN COMPLEX WITH CHEMICAL LIGAND Descriptor: BETA-SECRETASE 1, DIMETHYL SULFOXIDE, N-[3-[(4R)-2-azanylidene-5,5-bis(fluoranyl)-4-methyl-1,3-oxazinan-4-yl]-4-fluoranyl-phenyl]-5-cyano-pyridine-2-carboxamide, ... Authors: Banner, D.W, Kuglstatter, A, Benz, J, Stihle, M. Deposit date: 2013-02-08 Release date: 2013-05-01 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.74 Å) Cite: Beta-Secretase (Bace1) Inhibitors with High in Vivo Efficacy Suitable for Clinical Evaluation in Alzheimer'S Disease. J.Med.Chem., 56, 2013
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2013-02-08
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