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P21-activated kinase 1 in complex with a 4-azaindole inhibitor

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6b16
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P21-activated kinase 1 in complex with a 4-azaindole inhibitor Descriptor: N~4~-(5-cyclopropyl-1H-pyrazol-3-yl)-N~2~-[(1S)-1-(1H-pyrrolo[3,2-b]pyridin-5-yl)ethyl]pyrimidine-2,4-diamine, SULFATE ION, Serine/threonine-protein kinase PAK 1 Authors: Rouge, L, Wang, W. Deposit date: 2017-09-16 Release date: 2017-10-25 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.285 Å) Cite: Synthesis and evaluation of a series of 4-azaindole-containing p21-activated kinase-1 inhibitors. Bioorg. Med. Chem. Lett., 26, 2016
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2017-09-16
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