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Crystal structure of acetyltransferase Eis from Mycobacterium tuberculosis in complex with droperidol

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Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Crystal structure of acetyltransferase Eis from Mycobacterium tuberculosis in complex with droperidol Descriptor: 3-[1-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-2,3,4,5-tetrahydropyridin-4-yl]-1~{H}-benzimidazol-2-one, DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, ... Authors: Punetha, A, Garneau-Tsodikova, S, Tsodikov, O.V. Deposit date: 2020-05-28 Release date: 2021-06-02 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.15 Å) Cite: Structure-based design of haloperidol analogues as inhibitors of acetyltransferase Eis from Mycobacterium tuberculosis to overcome kanamycin resistance Rsc Med Chem, 12, 2021
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2020-05-28
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