遇见数据集

Jak3 with covalent inhibitor 4

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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Jak3 with covalent inhibitor 4 Descriptor: 1-{(3R)-3-[(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}propan-1-one, Tyrosine-protein kinase JAK3 Authors: Vajdos, F.F. Deposit date: 2016-11-04 Release date: 2017-02-22 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.34 Å) Cite: Design of a Janus Kinase 3 (JAK3) Specific Inhibitor 1-((2S,5R)-5-((7H-Pyrrolo[2,3-d]pyrimidin-4-yl)amino)-2-methylpiperidin-1-yl)prop-2-en-1-one (PF-06651600) Allowing for the Interrogation of JAK3 Signaling in Humans. J. Med. Chem., 60, 2017

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2016-11-04
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