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Toxoplasma gondii TS-DHFR in complex with selective inhibitor 3

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6n1t
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Toxoplasma gondii TS-DHFR in complex with selective inhibitor 3 Descriptor: 10-PROPARGYL-5,8-DIDEAZAFOLIC ACID, 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, 5-{4-[3-(2-methoxypyrimidin-5-yl)phenyl]piperazin-1-yl}pyrimidine-2,4-diamine, ... Authors: Hopper, A.T, Brockman, A, Wise, A, Gould, J, Barks, J, Radke, J.B, Sibley, L.D, Zou, Y, Thomas, S.B. Deposit date: 2018-11-11 Release date: 2019-01-23 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (3.5 Å) Cite: Discovery of Selective Toxoplasma gondii Dihydrofolate Reductase Inhibitors for the Treatment of Toxoplasmosis. J. Med. Chem., 62, 2019
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2018-11-11
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