Retinoic acid receptor-related orphan receptor (ROR) gamma in complex with allosteric compound 28
收藏Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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Retinoic acid receptor-related orphan receptor (ROR) gamma in complex with allosteric compound 28 Descriptor: (3S,4R)-1-[1-(2-chloro-6-cyclopropylbenzene-1-carbonyl)-4-fluoro-1H-indazol-3-yl]-3-hydroxypiperidine-4-carboxylic acid, Nuclear receptor ROR-gamma Authors: Palte, R.L, Parthasarathy, G. Deposit date: 2019-09-16 Release date: 2020-03-04 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.87 Å) Cite: Discovery ofN-(Indazol-3-yl)piperidine-4-carboxylic Acids as ROR gamma t Allosteric Inhibitors for Autoimmune Diseases. Acs Med.Chem.Lett., 11, 2020
创建时间:
2019-09-16



