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Crystal structure of the p300 acetyltransferase domain with AcCoA competitive inhibitor 17

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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Crystal structure of the p300 acetyltransferase domain with AcCoA competitive inhibitor 17 Descriptor: (2R)-2-{[(2S)-2-(4-cyanophenyl)propyl]amino}-N-[5-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-2-phenylacetamide, CHLORIDE ION, Histone acetyltransferase p300, ... Authors: Gardberg, A.S, Wilson, J.E. Deposit date: 2019-12-11 Release date: 2020-04-01 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Early Drug-Discovery Efforts towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors. Chemmedchem, 15, 2020
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2019-12-11
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