Structure of TTBK1 kinase domain in complex with Compound 3
收藏Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Structure of TTBK1 kinase domain in complex with Compound 3 Descriptor: 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol, SODIUM ION, Tau-tubulin kinase 1 Authors: Chodaprambil, J.V. Deposit date: 2020-08-28 Release date: 2021-05-19 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.56 Å) Cite: Discovery of Potent and Brain-Penetrant Tau Tubulin Kinase 1 (TTBK1) Inhibitors that Lower Tau Phosphorylation In Vivo. J.Med.Chem., 64, 2021
创建时间:
2020-08-28



