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Engineered RabGGTase in complex with BMS analogue 12

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Protein Data Bank Japan2023-11-08 更新2026-03-21 收录
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Engineered RabGGTase in complex with BMS analogue 12 Descriptor: 4-({(3R)-7-cyano-4-[(4-methoxyphenyl)sulfonyl]-1-[(1-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl}methyl)phenyl benzylcarbamate, CALCIUM ION, Geranylgeranyl transferase type-2 subunit alpha, ... Authors: Guo, Z, Stigter, E.A, Bon, R.S, Waldmann, H, Blankenfeldt, W, Goody, R.S. Deposit date: 2012-08-29 Release date: 2012-10-24 Last modified: 2023-11-08 Method: X-RAY DIFFRACTION (2.05 Å) Cite: Development of Selective, Potent RabGGTase Inhibitors J.Med.Chem., 55, 2012
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2012-08-29
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