KRasG12C ligand complex
收藏Protein Data Bank Japan2025-10-01 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/6t5v
下载链接
链接失效反馈官方服务:
资源简介:
KRasG12C ligand complex Descriptor: 1-[4-[6-chloranyl-7-(5-methyl-1~{H}-indazol-4-yl)quinazolin-4-yl]piperazin-1-yl]propan-1-one, GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, ... Authors: Phillips, C. Deposit date: 2019-10-17 Release date: 2020-02-19 Last modified: 2025-10-01 Method: X-RAY DIFFRACTION (1.31 Å) Cite: Structure-Based Design and Pharmacokinetic Optimization of Covalent Allosteric Inhibitors of the Mutant GTPase KRASG12C. J.Med.Chem., 63, 2020
创建时间:
2019-10-17



