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RORgamma in complex with inverse agonist 16

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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RORgamma in complex with inverse agonist 16 Descriptor: 4-chloro-3-[1-(2-chloro-6-fluorobenzoyl)-1,2,3,4-tetrahydroquinolin-6-yl]-N-methylbenzamide, Nuclear receptor ROR-gamma Authors: Marcotte, D.J. Deposit date: 2015-04-29 Release date: 2015-06-17 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.5 Å) Cite: Discovery of biaryl carboxylamides as potent ROR gamma inverse agonists. Bioorg.Med.Chem.Lett., 25, 2015

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2015-04-29
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