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Crystal structure of MLLT1 (ENL) YEATS domain in complexed with piperazine-urea derivative 1

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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Crystal structure of MLLT1 (ENL) YEATS domain in complexed with piperazine-urea derivative 1 Descriptor: 1,2-ETHANEDIOL, 4-(4-ethanoylphenyl)-~{N}-[(6-methoxypyridin-3-yl)methyl]piperazine-1-carboxamide, Protein ENL Authors: Chaikuad, A, Heidenreich, D, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Fedorov, O, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2019-10-04 Release date: 2019-11-06 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Structural Insights into Interaction Mechanisms of Alternative Piperazine-urea YEATS Domain Binders in MLLT1. Acs Med.Chem.Lett., 10, 2019
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2019-10-04
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