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hDHFR-OAG binary complex

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Protein Data Bank Japan2023-09-13 更新2026-03-21 收录
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hDHFR-OAG binary complex Descriptor: 6-{[(2,5-dichlorophenyl)amino]methyl}pyrido[2,3-d]pyrimidine-2,4-diamine, Dihydrofolate reductase, SULFATE ION Authors: Cody, V, Pace, J, Queener, S, Adair, O, Gangjee, A. Deposit date: 2012-07-23 Release date: 2014-01-29 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (1.35 Å) Cite: Kinetic and structural analysis for potent antifolate inhibition of Pneumocystis jirovecii, Pneumocystis carinii, and human dihydrofolate reductases and their active-site variants. Antimicrob.Agents Chemother., 57, 2013
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2012-07-23
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