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Cys-42-tethered stabilizer 12 of 14-3-3(sigma)/ERa PPI

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Cys-42-tethered stabilizer 12 of 14-3-3(sigma)/ERa PPI Descriptor: 14-3-3 protein sigma, 2-(4-bromanyl-3-methoxy-phenoxy)-2-methyl-~{N}-(2-sulfanylethyl)propanamide, Estrogen receptor, ... Authors: Sijbesma, E, Ottmann, C. Deposit date: 2020-12-15 Release date: 2021-07-07 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.1 Å) Cite: Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers. Acs Med.Chem.Lett., 12, 2021
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2020-12-15
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