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Crystal structure of human Bromodomain-containing protein 4 (BRD4) bromodomain with MS645

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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Crystal structure of human Bromodomain-containing protein 4 (BRD4) bromodomain with MS645 Descriptor: 1,2-ETHANEDIOL, Bromodomain-containing protein 4, N,N'-(decane-1,10-diyl)bis{2-[(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetamide} Authors: Ren, C, Zhou, M.M. Deposit date: 2018-05-25 Release date: 2018-07-25 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (1.46 Å) Cite: Spatially constrained tandem bromodomain inhibition bolsters sustained repression of BRD4 transcriptional activity for TNBC cell growth. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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2018-05-25
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