Crystal structure of pregnane X receptor ligand binding domain complexed with T0901317 analog T0-C6
收藏Protein Data Bank Japan2023-10-25 更新2026-04-19 收录
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Crystal structure of pregnane X receptor ligand binding domain complexed with T0901317 analog T0-C6 Descriptor: N-[4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenyl]-N-hexylbenzenesulfonamide, Nuclear receptor subfamily 1 group I member 2 Authors: Huber, A.D, Poudel, S, Seetharaman, J, Miller, D.J, Lin, W, Li, Y, Chen, T. Deposit date: 2022-10-11 Release date: 2023-03-15 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (2.37 Å) Cite: Structure-guided approach to modulate small molecule binding to a promiscuous ligand-activated protein. Proc.Natl.Acad.Sci.USA, 120, 2023
创建时间:
2022-10-11



