MELK in complex with NVS-MELK8A
收藏Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5ih9
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MELK in complex with NVS-MELK8A Descriptor: 1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1H-pyrazol-1-yl)phenyl]piperazine, Maternal embryonic leucine zipper kinase Authors: Sprague, E.R, Puleo, D.E. Deposit date: 2016-02-29 Release date: 2016-06-01 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (1.79 Å) Cite: Toward the Validation of Maternal Embryonic Leucine Zipper Kinase: Discovery, Optimization of Highly Potent and Selective Inhibitors, and Preliminary Biology Insight. J.Med.Chem., 59, 2016
创建时间:
2016-02-29



